A new and simple method for the synthesis of highly functionalised pyrrolizidines, indolizidines and pyrroloazepines

Paul A. O'Gorman, Ting Chen, Hannah E. Cross, Saleena Naeem, Arnaud Pitard, M. Ilyas Qamar, Karl Hemming

Research output: Contribution to journalArticle

15 Citations (Scopus)

Abstract

The reaction of 5-, 6- and 7-membered cyclic thioimidates with cyclopropenones gives access to highly functionalised pyrrolizidines, indolizidines and pyrroloazepines via a formal [3+2] cycloaddition process.

LanguageEnglish
Pages6316-6319
Number of pages4
JournalTetrahedron Letters
Volume49
Issue number44
Early online date23 Aug 2008
DOIs
Publication statusPublished - 27 Oct 2008

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Indolizidines
Cycloaddition
Cycloaddition Reaction
cyclopropenone

Cite this

O'Gorman, Paul A. ; Chen, Ting ; Cross, Hannah E. ; Naeem, Saleena ; Pitard, Arnaud ; Qamar, M. Ilyas ; Hemming, Karl. / A new and simple method for the synthesis of highly functionalised pyrrolizidines, indolizidines and pyrroloazepines. In: Tetrahedron Letters. 2008 ; Vol. 49, No. 44. pp. 6316-6319.
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A new and simple method for the synthesis of highly functionalised pyrrolizidines, indolizidines and pyrroloazepines. / O'Gorman, Paul A.; Chen, Ting; Cross, Hannah E.; Naeem, Saleena; Pitard, Arnaud; Qamar, M. Ilyas; Hemming, Karl.

In: Tetrahedron Letters, Vol. 49, No. 44, 27.10.2008, p. 6316-6319.

Research output: Contribution to journalArticle

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AU - Cross, Hannah E.

AU - Naeem, Saleena

AU - Pitard, Arnaud

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AU - Hemming, Karl

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